Cat No:LP000056 Product Name: GSK1904529A CAS NO:1089283-49-7 Molecular Formula:C44H47F2N9O5S Molecular Weight:851.96300 Purity: ≥98% Solubility: In DMSO Storage: -10°C GSK1904529A is a selective inhibitor of IGF-1R and IR with IC50 of 27 nM and 25 nM, >100-fold more selective for IGF-1R/InsR than Akt1/2, Aurora A/B,B-Raf, CDK2, EGFR etc. IC50 value: 27/25 nM (IGF1R/IR) [1] Target: IGF1R/IR […]
Cat No:LP000055 Product Name: Telatinib,BAY 57-9352 CAS NO:332012-40-5 Molecular Formula:C20H16ClN5O3 Molecular Weight:409.82600 Purity: ≥98% Solubility: In DMSO Storage: -10°C Telatinib has low affinity for the Raf kinase pathway, epidermal growth factor receptor family, the fibroblast growth factor receptor (FGFR) family, or the Tie-2 receptor[2]. Telatinib is metabolized by various cytochrome P450 (CYP) isoforms including CYP3A4/3A5, […]