Canetinib

Active small molecule, Products, , ,

Cat No:LP000124 Product Name:Canetinib;CI-1033;PD-183805 CAS No:267243-28-7 Purity: ≥99% Solubility: In DMSO Storage: -10°C Canertinib significantly inhibits growth of cultured melanoma cells, RaH3 and RaH5, in a dose-dependent manner. IC50 is approximately 0.8 μM and by 5μM both cell lines are completely growth-arrested within 72 h of treatment. Incubation of exponentially growing RaH3 and RaH5 with […]

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Ciproxifan

Active small molecule, Products, ,

Cat No:LP000123 Product Name:Ciproxifan;FUB359 CAS No:184025-18-1 Purity: ≥99% Solubility: In DMSO Storage: -10°C Ciproxifan(FUB-359) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at other receptor subtypes. IC50 value: 9.2 nM(Ki) Target: H3 receptor In vitro, Ciproxifan behaved as a competitive antagonist at the H3 autoreceptor […]

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