Cat No:LP000136 Product Name:OC000459;Timapiprant CAS No:851723-84-7 Purity: ≥99% Solubility: In DMSO Storage: -10°C OC000459 is a potent and selective D prostanoid receptor 2 (DP2) antagonist with IC50 of 13 nM. IC50 Value: 13 nM( Ki for hrCRTH2); 3 nM( Ki for Rat rCRTH2);13 nM(Ki for human native CRTH2) Target: D prostanoid receptor 2 CRTH2 (chemoattractant […]
Cat No:LP000135 Product Name:ARN-509 CAS No:956104-40-8 Purity: ≥99% Solubility: In DMSO Storage: -10°C ARN-509 also exhibits low micromolar affinity (IC50 3 μM) for the GABAA receptor in radioligand binding-assays and thus may potentially antagonize GABAA at therapeutic dose levels[1]. Apalutamide is a potent androgen receptor (AR) antagonist that targets the AR ligand-binding domain and prevents […]