Lersivirine(UK 453061)

Active small molecule, Products,

Cat No:LP000206 Product Name:Lersivirine,UK 453061 CAS No:473921-12-9 Purity: ≥99% Solubility: In DMSO Storage: -10°C Lersivirine(UK-453061) is a next-generation non-nucleoside reverse transcriptase inhibitor (NNRTI, IC50=119 nM) with a unique resistance profile that exhibits potent antiretroviral activity against wild-type human immunodeficiency virus and clinically relevant NNRTI-resistant strains. IC50 value: 0.119 uM [1] Target: NNRTI UK-453061(Compound 5) demonstrated […]

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Dabigatran etexilate mesylate

Active small molecule, Products, , ,

Cat No:LP000205 Product Name:Dabigatran etexilate mesylate;Pradaxa;BIBR 1048MS CAS No:872728-81-9 Purity: ≥99% Solubility: In DMSO Storage: -10°C Dabigatran etexilate mesylate (BIBR 1048MS) is the orally active prodrug of dabigatran. Dabigatran is a reversible and selective, direct thrombin inhibitor (DTI) with Ki value of 4.5 nM. IC50 Value: 4.5 nM (Ki); 10 nM(Thrombin-induced platelet aggregation) [1] in […]

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