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Guanoclor

Jul 17, 2018adminActive small molecule, Products5001-32-1, Guanoclor, VATENSOL

Cat No:LP000416 Product Name:Guanoclor;VATENSOL CAS#5001-32-1 Molecular Formula:C9H12Cl2N4O Molecular Weight：263.13

EPZ011989

Jul 17, 2018adminActive small molecule, Products1598383-40-4, EPZ011989

Cat No:LP000415 Product Name:EPZ011989 CAS#1598383-40-4 EPZ011989 is a potent, selective orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 wt and EZH2 Y646; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase. IC50 value: < 3 nM ( Ki for wt EZH2, EZH2 Y646) Target: EZH2 inhibitor In vitro: EPZ011989 is also […]