| Name | N-[(1,2-Dihydro-4,6-dimethyl-2-oxo-3-pyridinyl)methyl]-5-[ethyl(tetrahydro-2H-pyran-4-yl)amino]-4-methyl-4′-(4-morpholinylmethyl)-[1,1′-biphenyl]-3-carboxamide | |
| Molecular Structure | ![CAS # 1403254-99-8, N-[(1,2-Dihydro-4,6-dimethyl-2-oxo-3-pyridinyl)methyl]-5-[ethyl(tetrahydro-2H-pyran-4-yl)amino]-4-methyl-4'-(4-morpholinylmethyl)-[1,1'-biphenyl]-3-carboxamide](https://www.chemblink.com/structures/1403254-99-8.gif) |
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| Molecular Formula | C34H44N4O4 | |
| Molecular Weight | 572.74 | |
| CAS Registry Number | 1403254-99-8 | |
EPZ-6438 (Tazemetostat)是一种有效，选择性，口服的 EZH2 抑制剂，Ki 和 IC50 分别为2.5和11 nM。